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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T0242L | Sitagliptin phosphate monohydrate | MK-0431,MK-0431 phosphate monohydrate | Proteasome , DPP-4 , Autophagy |
T23358 | Sitagliptin phosphate | Januvia,MK-0431 phosphate,Sitagliptin (phosphate) | DPP-4 , Autophagy |
Sitagliptin phosphate (MK-0431 phosphate) is a dipeptidyl peptidase-4 (DPP4) inhibitor. | |||
T40930 | (S)-Sitagliptin phosphate | (S)-Sitagliptin phosphate,(S)-MK-0431 phosphate | |
(S)-Sitagliptin phosphate, the less active S-enantiomer of Sitagliptin phosphate, is a high-potency inhibitor of DPP4. It exhibits an IC50 of 19 nM in Caco-2 cell extracts. |